Reaction assignment
RHEA:10748CA6 · RHEA:10748 assignment
Protein-specific UniProt catalytic-activity assignment joined to a balanced Rhea master reaction.
Open the recordEvidence records
Release haca-evidence-v1-4bf3e75a91408390. 120 evidence records: 80 experimental structure mappings, 28 direct assay activities and 12 protein-specific reaction assignments. Each record lists every source it came from and, for measurements, the value exactly as the source reported it.
120 evidence records in this view, page 5 of 5.
Assay activity
2456868CA7 · ChEMBL activity 2456868
Kinact source measurement: = 5.73 uM. No cross-assay comparison is prequalified.
Not comparable: CONDITION_MISSING
Open the recordAssay activity
2619680CA7 · ChEMBL activity 2619680
Ki source measurement: = 5.1 nM. No cross-assay comparison is prequalified.
Not comparable: CONDITION_MISSING
Open the recordExperimental structure
3MDZCA7 · PDB 3MDZ
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
3ML5CA7 · PDB 3ML5
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6G4TCA7 · PDB 6G4T
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6H36CA7 · PDB 6H36
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6H37CA7 · PDB 6H37
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6H38CA7 · PDB 6H38
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6ZR9CA7 · PDB 6ZR9
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
8Q3UCA7 · PDB 8Q3U
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordReaction assignment
RHEA:10748CA7 · RHEA:10748 assignment
Protein-specific UniProt catalytic-activity assignment joined to a balanced Rhea master reaction.
Open the recordExperimental structure
2W2JCA8 · PDB 2W2J
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordAssay activity
2393967CA9 · ChEMBL activity 2393967
Ki source measurement: = 1.84 uM. No cross-assay comparison is prequalified.
Not comparable: CONDITION_MISSING
Open the recordAssay activity
2598328CA9 · ChEMBL activity 2598328
Ki source measurement: = 26.0 nM. No cross-assay comparison is prequalified.
Not comparable: CONDITION_MISSING
Open the recordExperimental structure
2HKFCA9 · PDB 2HKF
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
3IAICA9 · PDB 3IAI
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
5DVXCA9 · PDB 5DVX
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
5FL4CA9 · PDB 5FL4
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
5FL6CA9 · PDB 5FL6
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6RQQCA9 · PDB 6RQQ
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
6RQUCA9 · PDB 6RQU
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordExperimental structure
8Q19CA9 · PDB 8Q19
X-ray diffraction structure mapped through PDBe/SIFTS.
Open the recordReaction assignment
RHEA:10748CA9 · RHEA:10748 assignment
Protein-specific UniProt catalytic-activity assignment joined to a balanced Rhea master reaction.
Open the record